compound 9 [PMID: 26937601] [Ligand Id: 9197] activity data from GtoPdb

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  • beta-secretase 1 in Human [GtoPdb: 2330] [UniProtKB: P56817]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
beta-secretase 1 in Human [GtoPdb: 2330] [UniProtKB: P56817]
GtoPdb Inhibition of recombinant hBACE1 by FRET assay; substrate QSY7EISEVNLDAEFC-Eu-amide - 8.3 pKi 5 nM Ki J Med Chem (2016) 59: 3231-48 [PMID:26937601]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.