CCT245737 [Ligand Id: 9187] activity data from GtoPdb

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  • checkpoint kinase 1 in Human [GtoPdb: 1987] [UniProtKB: O14757]
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  • checkpoint kinase 2 in Human [GtoPdb: 1988] [UniProtKB: O96017]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
checkpoint kinase 1 in Human [GtoPdb: 1987] [UniProtKB: O14757]
GtoPdb - - 8.89 pIC50 1.3 nM IC50 J Med Chem (2016) 59: 5221-37 [PMID:27167172]
checkpoint kinase 2 in Human [GtoPdb: 1988] [UniProtKB: O96017]
GtoPdb - - 5.61 pIC50 2440 nM IC50 J Med Chem (2016) 59: 5221-37 [PMID:27167172]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.