BAY-524 [Ligand Id: 9127] activity data from GtoPdb

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  • BUB1 mitotic checkpoint serine/threonine kinase in Human [GtoPdb: 1949] [UniProtKB: O43683]
Created with Highcharts 10.3.3ValuesChart context menuBUB1 mitotic checkpoint serine/threonine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BUB1 mitotic checkpoint serine/threonine kinase in Human [GtoPdb: 1949] [UniProtKB: O43683]
GtoPdb Measuring inhibition of the recombinant catalytic domain of human Bub1 (amino acids 704–1085). - 6.35 pIC50 450 nM IC50 Elife (2016) 5: [PMID:26885717]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.