(R)-ARN2508 [Ligand Id: 9000] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| COX-1 in Human [GtoPdb: 1375] [UniProtKB: P23219] | ||||||||
| GtoPdb | - | - | 5.4 | pIC50 | 4000 | nM | IC50 | Eur J Med Chem (2016) 109: 216-37 [PMID:26774927] |
| COX-2 in Human [GtoPdb: 1376] [UniProtKB: P35354] | ||||||||
| GtoPdb | - | - | 4.64 | pIC50 | 22800 | nM | IC50 | Eur J Med Chem (2016) 109: 216-37 [PMID:26774927] |
| Fatty acid amide hydrolase in Human [GtoPdb: 1400] [UniProtKB: O00519] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | 9.9 | nM | IC50 | Eur J Med Chem (2016) 109: 216-37 [PMID:26774927] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
