MS023 [Ligand Id: 8955] activity data from GtoPdb

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  • protein arginine methyltransferase 1 in Human [GtoPdb: 1252] [UniProtKB: Q99873]
Created with Highcharts 10.3.3ValuesChart context menuprotein arginine methyltransferase 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • protein arginine methyltransferase 3 in Human [GtoPdb: 1254] [UniProtKB: O60678]
Created with Highcharts 10.3.3ValuesChart context menuprotein arginine methyltransferase 3pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
Created with Highcharts 10.3.3ValuesChart context menucoactivator associated arginine methyltransferase 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • protein arginine methyltransferase 6 in Human [GtoPdb: 1257] [UniProtKB: Q96LA8]
Created with Highcharts 10.3.3ValuesChart context menuprotein arginine methyltransferase 6pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • protein arginine methyltransferase 8 in Human [GtoPdb: 1259] [UniProtKB: Q9NR22]
Created with Highcharts 10.3.3ValuesChart context menuprotein arginine methyltransferase 8pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
protein arginine methyltransferase 1 in Human [GtoPdb: 1252] [UniProtKB: Q99873]
GtoPdb - - 7.96 pKi 11 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 3 in Human [GtoPdb: 1254] [UniProtKB: O60678]
GtoPdb - - 7.26 pKi 55 nM Ki ACS Chemical Biology (2015) :
coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
GtoPdb - - 7.64 pKi 23 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 6 in Human [GtoPdb: 1257] [UniProtKB: Q96LA8]
GtoPdb - - 8.22 pKd 6 nM Kd ACS Chemical Biology (2015) :
GtoPdb - - 9.1 pKi 0.8 nM Ki ACS Chemical Biology (2015) :
protein arginine methyltransferase 8 in Human [GtoPdb: 1259] [UniProtKB: Q9NR22]
GtoPdb - - 8.89 pKi 1.3 nM Ki ACS Chemical Biology (2015) :

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.