fimepinostat [Ligand Id: 8952] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
| GtoPdb | - | - | 7.72 | pIC50 | 19 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | - | - | 7.27 | pIC50 | 54 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
| GtoPdb | - | - | 7.41 | pIC50 | 39 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
| GtoPdb | - | - | 6.51 | pIC50 | 311 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 10 in Human [GtoPdb: 2614] [UniProtKB: Q969S8] | ||||||||
| GtoPdb | - | - | 8.55 | pIC50 | 2.8 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 11 in Human [GtoPdb: 2615] [UniProtKB: Q96DB2] | ||||||||
| GtoPdb | - | - | 8.27 | pIC50 | 5.4 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 2 in Human [GtoPdb: 2616] [UniProtKB: Q92769] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | 5 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379] | ||||||||
| GtoPdb | - | - | 8.74 | pIC50 | 1.8 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 6 in Human [GtoPdb: 2618] [UniProtKB: Q9UBN7] | ||||||||
| GtoPdb | - | - | 7.57 | pIC50 | 27 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
| histone deacetylase 1 in Human [GtoPdb: 2658] [UniProtKB: Q13547] | ||||||||
| GtoPdb | - | - | 8.77 | pIC50 | 1.7 | nM | IC50 | Clin Cancer Res (2012) 18: 4104-13 [PMID:22693356] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
