compound 16 [PMID: 19097778] [Ligand Id: 8837] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL482331
  • Solute carrier family 28 member 3 in Human [ChEMBL: CHEMBL5707] [GtoPdb: 1116] [UniProtKB: Q9HAS3]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Solute carrier family 28 member 3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5707] [GtoPdb: 1116] [UniProtKB: Q9HAS3]
GtoPdb - - 5.54 pKi 2880 nM Ki Bioorg Med Chem Lett (2009) 19: 917-21 [PMID:19097778]
ChEMBL Binding affinity to human recombinant CNT3 expressed in pig PK15NTD cells assessed as [3H]uridine uptake by beta-scintillation counter B 5.54 pKi 2880 nM Ki Bioorg Med Chem Lett (2009) 19: 917-921 [PMID:19097778]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]