Cy3B-telenzepine [Ligand Id: 8598] activity data from GtoPdb

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  • M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229]
Created with Highcharts 10.3.3ValuesChart context menuM1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172]
Created with Highcharts 10.3.3ValuesChart context menuM2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229]
GtoPdb - - 10.5 pKd - - - Proc Natl Acad Sci USA (2010) 107: 2693-8 [PMID:20133736]
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172]
GtoPdb - - 10.4 pKi - - - J Mol Cell Cardiol (2013) 57: 129-36 [PMID:23357106]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.