Ro5028442 [Ligand Id: 8529] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288] | ||||||||
| GtoPdb | - | - | 9 | pKi | 1 | nM | Ki | J Med Chem (2015) 58: 2275-89 [PMID:25654260] |
| V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518] | ||||||||
| GtoPdb | - | - | 4.52 | pKi | >30000 | nM | Ki | J Med Chem (2015) 58: 2275-89 [PMID:25654260] |
| OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559] | ||||||||
| GtoPdb | - | - | 5 | pKi | 9891 | nM | Ki | J Med Chem (2015) 58: 2275-89 [PMID:25654260] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
