compound 58 [PMID: 25037917] [Ligand Id: 8520] activity data from GtoPdb

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  • DAT in Human [GtoPdb: 927] [UniProtKB: Q01959]
Created with Highcharts 10.3.3ValuesChart context menuDATpKd HumanpKi HumanpIC50 HumanpEC50 Human0123456Highcharts.com
  • PROT in Human [GtoPdb: 938] [UniProtKB: Q99884]
Created with Highcharts 10.3.3ValuesChart context menuPROTpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
DAT in Human [GtoPdb: 927] [UniProtKB: Q01959]
GtoPdb - - 5.21 pIC50 6100 nM IC50 Bioorg Med Chem Lett (2014) 24: 3886-90 [PMID:25037917]
PROT in Human [GtoPdb: 938] [UniProtKB: Q99884]
GtoPdb - - 7.74 pIC50 18 nM IC50 Bioorg Med Chem Lett (2014) 24: 3886-90 [PMID:25037917]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.