relenopride [Ligand Id: 8427] activity data from GtoPdb

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  • 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
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  • 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
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  • 5-HT4 receptor in Human [GtoPdb: 9] [UniProtKB: Q13639]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
GtoPdb - - 6.22 pKi 600 nM Ki Neurogastroenterol Motil (2014) 26: 1761-70 [PMID:25316608]
5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
GtoPdb - - 7.51 pKi 31 nM Ki Neurogastroenterol Motil (2014) 26: 1761-70 [PMID:25316608]
5-HT4 receptor in Human [GtoPdb: 9] [UniProtKB: Q13639]
GtoPdb - - 8.3 pKi 4.96 nM Ki Neurogastroenterol Motil (2014) 26: 1761-70 [PMID:25316608]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.