I-CBP112 [Ligand Id: 8236] activity data from GtoPdb

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  • CREB binding protein in Human [GtoPdb: 2734] [UniProtKB: Q92793]
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  • E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CREB binding protein in Human [GtoPdb: 2734] [UniProtKB: Q92793]
GtoPdb Isothermal titration calorimetry (ITC) assay. - 6.85 pKd 142 nM Kd I-CBP112 A CREBBP/EP300-selective chemical probe. thesgc.org
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb Isothermal titration calorimetry (ITC) assay. - 6.2 pKd 625 nM Kd I-CBP112 A CREBBP/EP300-selective chemical probe. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.