CRT 0066101 [Ligand Id: 8048] activity data from GtoPdb

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  • protein kinase D1 in Human [GtoPdb: 1489] [UniProtKB: Q15139]
Created with Highcharts 10.3.3ValuesChart context menuprotein kinase D1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • protein kinase D2 in Human [GtoPdb: 2173] [UniProtKB: Q9BZL6]
Created with Highcharts 10.3.3ValuesChart context menuprotein kinase D2pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • protein kinase D3 in Human [GtoPdb: 2174] [UniProtKB: O94806]
Created with Highcharts 10.3.3ValuesChart context menuprotein kinase D3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
protein kinase D1 in Human [GtoPdb: 1489] [UniProtKB: Q15139]
GtoPdb - - 9 pIC50 1 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]
protein kinase D2 in Human [GtoPdb: 2173] [UniProtKB: Q9BZL6]
GtoPdb - - 8.6 pIC50 2.5 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]
protein kinase D3 in Human [GtoPdb: 2174] [UniProtKB: O94806]
GtoPdb - - 8.7 pIC50 2 nM IC50 Mol Cancer Ther (2010) 9: 1136-46 [PMID:20442301]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.