riviciclib [Ligand Id: 7934] activity data from GtoPdb

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  • cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493]
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  • cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
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  • cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493]
GtoPdb CDK1/cyclin B complex - 7.1 pIC50 79 nM IC50 Mol Cancer Ther (2007) 6: 918-25 [PMID:17363486]
cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802]
GtoPdb CDK4/cyclin D1 complex - 7.2 pIC50 63 nM IC50 Mol Cancer Ther (2007) 6: 918-25 [PMID:17363486]
cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750]
GtoPdb CDK9/cyclin T1 complex - 7.7 pIC50 20 nM IC50 Mol Cancer Ther (2007) 6: 918-25 [PMID:17363486]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.