bitopertin [Ligand Id: 7546] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GlyT1 in Human [GtoPdb: 935] [UniProtKB: P48067] | ||||||||
| GtoPdb | - | - | 7.33 | pKi | 47 | nM | Ki | J Med Chem (2018) 61: 7503-7524 [PMID:30080045] |
| GtoPdb | - | - | 7.52 | pEC50 | 30 | nM | EC50 | J Med Chem (2010) 53: 4603-14 [PMID:20491477] |
| GlyT2 in Human [GtoPdb: 936] [UniProtKB: Q9Y345] | ||||||||
| GtoPdb | - | - | 4.52 | pEC50 | >30000 | nM | EC50 | J Med Chem (2010) 53: 4603-14 [PMID:20491477] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
