H3-CoA-20 [Ligand Id: 7035] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1221562
  • EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
Created with Highcharts 10.3.3ValuesChart context menuEP300 lysine acetyltransferasepKd HumanpKi HumanpIC50 HumanpEC50 Human01234Highcharts.com
  • lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
Created with Highcharts 10.3.3ValuesChart context menulysine acetyltransferase 2BpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 3.7 pIC50 200000 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
GtoPdb - - 6.52 pIC50 300 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]

ChEMBL data shown on this page come from version 35:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]