CTEP [Ligand Id: 6409] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mGlu5 receptor in Human [GtoPdb: 293] [UniProtKB: P41594] | ||||||||
| GtoPdb | - | - | 7.79 | pKi | 16.4 | nM | Ki |
J Pharmacol Exp Ther (2011) 339: 474-86 [PMID:21849627]; J Med Chem (2015) 58: 1358-71 [PMID:25565255] |
| GtoPdb | - | - | 8.19 | pIC50 | 6.4 | nM | IC50 | J Pharmacol Exp Ther (2011) 339: 474-86 [PMID:21849627] |
| mGlu5 receptor in Mouse [GtoPdb: 293] [UniProtKB: Q3UVX5] | ||||||||
| GtoPdb | - | - | 8.02 | pKi | 9.5 | nM | Ki | J Pharmacol Exp Ther (2011) 339: 474-86 [PMID:21849627] |
| mGlu5 receptor in Rat [GtoPdb: 293] [UniProtKB: P31424] | ||||||||
| GtoPdb | - | - | 7.9 | pKi | 12.6 | nM | Ki | J Pharmacol Exp Ther (2011) 339: 474-86 [PMID:21849627] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
