phenylacetyl-Ala,DTrp-phenthylamide [Ligand Id: 6192] activity data from GtoPdb

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  • BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
  • BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
  • BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
Created with Highcharts 10.3.3ValuesChart context menuBB3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 MousepKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
GtoPdb - - 5.5 pIC50 3162 nM IC50 Peptides (2010) 31: 1569-78 [PMID:20438784]
GtoPdb - - 8.92 pEC50 1.2 nM EC50 J Pept Sci (2002) 8: 461-75 [PMID:12212809];
Biochem Biophys Res Commun (2009) 387: 283-8 [PMID:19580790]
BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
GtoPdb - - 7.48 pEC50 33.3 nM EC50 Biochem Biophys Res Commun (2009) 387: 283-8 [PMID:19580790]
BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
GtoPdb - - 6.96 pEC50 109.9 nM EC50 Biochem Biophys Res Commun (2009) 387: 283-8 [PMID:19580790]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.