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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336] | ||||||||
| GtoPdb | - | - | 5.48 | pIC50 | 3300 | nM | IC50 |
Cell Metab (2010) 11: 101-12 [PMID:20096642]; Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571] |
| BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
| GtoPdb | - | - | 5.36 | pIC50 | 4400 | nM | IC50 |
Cell Metab (2010) 11: 101-12 [PMID:20096642]; Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571] |
| BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247] | ||||||||
| GtoPdb | - | - | 8.7 | pIC50 | 2 | nM | IC50 |
Cell Metab (2010) 11: 101-12 [PMID:20096642]; Pharmacol Exp Therap (2013) 347: 100-116 [PMID:23892571]; J Pharmacol Exp Ther (2019) 369: 454-465 [PMID:30971479] |
| BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798] | ||||||||
| GtoPdb | - | - | 8.09 | pIC50 | 8.1 | nM | IC50 | Cell Metab (2010) 11: 101-12 [PMID:20096642] |
| BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418] | ||||||||
| GtoPdb | - | - | 8.77 | pIC50 | 1.7 | nM | IC50 | Cell Metab (2010) 11: 101-12 [PMID:20096642] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.