gastrin-releasing peptide [Ligand Id: 612] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BB1 receptor in Rat [GtoPdb: 38] [UniProtKB: P24053] | ||||||||
| GtoPdb | - | - | 6.39 | pKi | 403 | nM | Ki |
J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496]; Mol Pharmacol (1995) 47: 10-20 [PMID:7838118]; J Biol Chem (1997) 272: 26062-71 [PMID:9325344]; Biochemistry (1999) 38: 7307-20 [PMID:10353842] |
| BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
| GtoPdb | - | - | 8.21 | pKi | 6.2 | nM | Ki |
J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496]; Mol Pharmacol (1995) 47: 10-20 [PMID:7838118]; Peptides (2011) 32: 1685-99 [PMID:21729729] |
| GtoPdb | - | - | 9.96 | pIC50 | 0.11 | nM | IC50 | Peptides (2009) 30: 1473-86 [PMID:19463875] |
| BB2 receptor in Mouse [GtoPdb: 39] [UniProtKB: P21729] | ||||||||
| GtoPdb | - | - | 8.91 | pKi | 1.24 | nM | Ki | Biochemistry (1999) 38: 7307-20 [PMID:10353842] |
| BB2 receptor in Rat [GtoPdb: 39] [UniProtKB: P52500] | ||||||||
| GtoPdb | - | - | 7.74 | pKi | 18 | nM | Ki |
Mol Pharmacol (1995) 47: 10-20 [PMID:7838118]; J Biol Chem (1997) 272: 26062-71 [PMID:9325344] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
