galmic [Ligand Id: 6119] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1187471 (Galmic) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| GAL1 receptor/Galanin receptor 1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4894] [GtoPdb: 243] [UniProtKB: P47211] | ||||||||
| ChEMBL | Binding affinity to human GalR1 | B | 4.47 | pKi | 34200 | nM | Ki | J Med Chem (2010) 53: 1871-1875 [PMID:20121116] |
| GtoPdb | - | - | 4.47 | pKi | 34200 | nM | Ki |
Neuropeptides (2005) 39: 161-3 [PMID:15944006]; Proc Natl Acad Sci USA (2004) 101: 10470-5 [PMID:15240875] |
| GAL2 receptor/Galanin receptor 2 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5577] [GtoPdb: 244] [UniProtKB: O08726] | ||||||||
| GtoPdb | - | - | 5 | pKd | >10000 | nM | Kd |
Proc Natl Acad Sci USA (2004) 101: 10470-5 [PMID:15240875]; Neuropeptides (2005) 39: 143-6 [PMID:15944002] |
| ChEMBL | Binding affinity to rat GalR2 | B | 4 | pKi | >100000 | nM | Ki | J Med Chem (2010) 53: 1871-1875 [PMID:20121116] |
ChEMBL data shown on this page come from version 34:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
