RO5166017 [Ligand Id: 5862] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| TA1 receptor in Human [GtoPdb: 364] [UniProtKB: Q96RJ0] | ||||||||
| GtoPdb | - | - | 7.5 | pKi | 31 | nM | Ki | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
| GtoPdb | - | - | 7.3 | pEC50 | 55 | nM | EC50 | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
| TA1 receptor in Mouse [GtoPdb: 364] [UniProtKB: Q923Y8] | ||||||||
| GtoPdb | - | - | 8.7 | pKi | 1.9 | nM | Ki | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
| GtoPdb | - | - | 8.5 | pEC50 | 3.3 | nM | EC50 | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
| TA1 receptor in Rat [GtoPdb: 364] [UniProtKB: Q923Y9] | ||||||||
| GtoPdb | - | - | 8.6 | pKi | 2.7 | nM | Ki | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
| GtoPdb | - | - | 7.9 | pEC50 | 14 | nM | EC50 | Proc Natl Acad Sci USA (2011) 108: 8485-90 [PMID:21525407] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
