1-oleoyl glycerol [Ligand Id: 5756] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL428593 (1-mono(cis-9-octacenoyl)glycerol, 1-monoolein, 1-monooleoyl-rac-glycerol, .alpha.-monoolein, FEMA NO. 2526, Glycerol 1-monooleate, Glycerol monooleate, Glyceryl 1-oleate, Glyceryl mono-oleate, Glyceryl monooleate, Glyceryl monooleate 40, Glyceryl monooleate 40%, Glyceryl monooleate 60, Glyceryl monooleate 90, Glyceryl monooleate 90%, Glyceryl oleate, Monolein, Mono-olein, Monoolein, NSC-406285, Olein, Rac-1-monooleoylglycerol) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| diacylglycerol kinase alpha/Diacylglycerol kinase alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4105787] [GtoPdb: 3256] [UniProtKB: P23743] | ||||||||
| ChEMBL | Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in presence of [gamma-32P]ATP | B | 4.04 | pKi | 91000 | nM | Ki | Eur J Med Chem (2019) 164: 378-390 [PMID:30611057] |
| GPR119 in Human [GtoPdb: 126] [UniProtKB: Q8TDV5] | ||||||||
| GtoPdb | - | - | 5.6 | pEC50 | - | - | - | J Clin Endocrinol Metab (2011) 96: E1409-17 [PMID:21778222] |
ChEMBL data shown on this page come from version 34:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
