MRS5151 [Ligand Id: 5622] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| A1 receptor in Human [GtoPdb: 18] [UniProtKB: P30542] | ||||||||
| GtoPdb | - | - | 4.83 | pKi | 14900 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
| A1 receptor in Mouse [GtoPdb: 18] [UniProtKB: Q60612] | ||||||||
| GtoPdb | - | - | 4.98 | pKi | 10500 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
| A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274] | ||||||||
| GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
| A2A receptor in Mouse [GtoPdb: 19] [UniProtKB: Q60613] | ||||||||
| GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
| A3 receptor in Human [GtoPdb: 21] [UniProtKB: P0DMS8] | ||||||||
| GtoPdb | - | - | 8.62 | pKi | 2.38 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
| A3 receptor in Mouse [GtoPdb: 21] [UniProtKB: Q61618] | ||||||||
| GtoPdb | - | - | 7.61 | pKi | 24.4 | nM | Ki | Bioorg Med Chem Lett (2008) 18: 2813-9 [PMID:18424135] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
