4-AMBA [Ligand Id: 4702] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL328875 (4-(Aminomethyl)Benzoic Acid, 4-Aminomethyl-Benzoic Acid, Aminomethylbenzoic acid)
  • Peptide transporter 1 in Human [GtoPdb: 984] [UniProtKB: P46059]
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  • Peptide transporter 2 in Human [GtoPdb: 985] [UniProtKB: Q16348]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Peptide transporter 1 in Human [GtoPdb: 984] [UniProtKB: P46059]
GtoPdb - - 2.3 pKi - - Ki J Nutr (2005) 135: 1491-5 [PMID:15930458];
J Physiol (Lond.) (1998) 512 ( Pt 3): 629-34 [PMID:9882198];
J Pharmacol Exp Ther (2010) 332: 220-8 [PMID:19789362]
Peptide transporter 2 in Human [GtoPdb: 985] [UniProtKB: Q16348]
GtoPdb - - 2.5 pKi - - - Amino Acids (2006) 31: 137-56 [PMID:16868651];
J Biol Chem (2002) 277: 7287-92 [PMID:11751927]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]