[3H]GlySar [Ligand Id: 4659] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL175737 (Glycylsarcosine, Gly-Sar, Gly-Sarcosin)
  • Peptide transporter 2/Solute carrier family 15 member 2 in Human [ChEMBL: CHEMBL1743125] [GtoPdb: 985] [UniProtKB: Q16348]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Peptide transporter 2/Solute carrier family 15 member 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1743125] [GtoPdb: 985] [UniProtKB: Q16348]
ChEMBL TP_TRANSPORTER: inhibition of Cephalexin uptake in SKPT cells F 4.19 pKi 64000 nM Ki J Biol Chem (1995) 270: 25672-25677 [PMID:7592745]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]