9-phenanthrol [Ligand Id: 4114] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL2407182 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| TRPM4/Transient receptor potential cation channel subfamily M member 4 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1628469] [GtoPdb: 496] [UniProtKB: Q8TD43] | ||||||||
| ChEMBL | Inhibition of TRPM4 (unknown origin) | B | 4.54 | pIC50 | 29000 | nM | IC50 | Eur J Med Chem (2019) 166: 167-177 [PMID:30708257] |
| GtoPdb | - | - | 4.78 | pIC50 | 16700 | nM | IC50 | Br J Pharmacol (2008) 153: 1697-705 [PMID:18297105] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
