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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229] | ||||||||
| GtoPdb | - | - | 7.1 | pKi | - | - | - | FEBS Lett (1994) 352: 91-4 [PMID:7925952] |
| M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172] | ||||||||
| GtoPdb | - | - | 6 | pKi | - | - | - | FEBS Lett (1994) 352: 91-4 [PMID:7925952] |
| GtoPdb | - | - | 6.3 | pA2 | - | - | - | J Pharmacol Exp Ther (1999) 288: 164-70 [PMID:9862767] |
| M3 receptor in Human [GtoPdb: 15] [UniProtKB: P20309] | ||||||||
| GtoPdb | - | - | 6 | pKi | - | - | - | FEBS Lett (1994) 352: 91-4 [PMID:7925952] |
| M4 receptor in Human [GtoPdb: 16] [UniProtKB: P08173] | ||||||||
| GtoPdb | - | - | 8.52 | pKi | 3 | nM | Ki | Invest Ophthalmol Vis Sci (2018) 59: 2778-2791 [PMID:29860464] |
| GtoPdb | - | - | 8.7 | pKi | - | - | - |
FEBS Lett (1994) 352: 91-4 [PMID:7925952]; J Pharmacol Exp Ther (1999) 288: 164-70 [PMID:9862767] |
| M5 receptor in Human [GtoPdb: 17] [UniProtKB: P08912] | ||||||||
| GtoPdb | - | - | 6 | pKi | - | - | - | FEBS Lett (1994) 352: 91-4 [PMID:7925952] |
| α2A-adrenoceptor in Human [GtoPdb: 25] [UniProtKB: P08913] | ||||||||
| GtoPdb | - | - | 8.3 | pKi | 5 | nM | Ki | Invest Ophthalmol Vis Sci (2018) 59: 2778-2791 [PMID:29860464] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.