AM966 [Ligand Id: 2905] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| LPA4 receptor in Human [GtoPdb: 94] [UniProtKB: Q99677] | ||||||||
| GtoPdb | - | - | 5.1 | pIC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
| LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633] | ||||||||
| GtoPdb | - | - | 7.8 | pIC50 | 15.8 | nM | IC50 | J Pharmacol Exp Ther (2011) 336: 693-700 [PMID:21159750] |
| LPA1 receptor in Mouse [GtoPdb: 272] [UniProtKB: P61793] | ||||||||
| GtoPdb | - | - | 7.7 | pEC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
| LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0] | ||||||||
| GtoPdb | - | - | 5.8 | pIC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
| LPA2 receptor in Mouse [GtoPdb: 273] [UniProtKB: Q9JL06] | ||||||||
| GtoPdb | - | - | 4.6 | pIC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
| LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5] | ||||||||
| GtoPdb | - | - | 5.7 | pIC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
| LPA3 receptor in Mouse [GtoPdb: 274] [UniProtKB: Q9EQ31] | ||||||||
| GtoPdb | - | - | 6.8 | pIC50 | - | - | - | Br J Pharmacol (2010) 160: 1699-713 [PMID:20649573] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
