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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Cav1.2 in Human [GtoPdb: 529] [UniProtKB: Q13936] | ||||||||
| GtoPdb | - | - | 6.4 | pIC50 | - | - | - | Mol Pharmacol (2002) 62: 1418-30 [PMID:12435810] |
| Cav2.2 in Human [GtoPdb: 533] [UniProtKB: Q00975] | ||||||||
| GtoPdb | - | - | 5.9 | pIC50 | - | - | - | Mol Pharmacol (2002) 62: 1418-30 [PMID:12435810] |
| Cav2.3 in Human [GtoPdb: 534] [UniProtKB: Q15878] | ||||||||
| GtoPdb | - | - | 7 | pIC50 | - | - | - | Mol Pharmacol (2002) 62: 1418-30 [PMID:12435810] |
| ASIC1 in Human [GtoPdb: 684] [UniProtKB: P78348] | ||||||||
| GtoPdb | - | - | 5.4 | pIC50 | ~4000 | nM | IC50 | J Biol Chem (2006) 281: 2497-505 [PMID:16319075] |
| GtoPdb | - | - | 5.8 | pIC50 | ~1500 | nM | IC50 | |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.