(-)-(R)-efonidipine [Ligand Id: 2519] activity data from GtoPdb

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  • Cav1.2 in Rat [GtoPdb: 529] [UniProtKB: P22002]
Created with Highcharts 10.3.3ValuesChart context menuCav1.2pKd RatpKi RatpIC50 RatpEC50 Rat01234Highcharts.com
  • Cav3.1 in Rat [GtoPdb: 535] [UniProtKB: O54898]
Created with Highcharts 10.3.3ValuesChart context menuCav3.1pKd RatpKi RatpIC50 RatpEC50 Rat02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Cav1.2 in Rat [GtoPdb: 529] [UniProtKB: P22002]
GtoPdb - - 3.5 pIC50 - - - Br J Pharmacol (2004) 143: 1050-7 [PMID:15545287]
Cav3.1 in Rat [GtoPdb: 535] [UniProtKB: O54898]
GtoPdb - - 7 pIC50 - - - Br J Pharmacol (2004) 143: 1050-7 [PMID:15545287]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.