[3H]RS 57639 [Ligand Id: 239] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1908857
  • 5-HT4 receptor in Rat [GtoPdb: 9] [UniProtKB: Q62758]
  • 5-HT4 receptor in Guinea pig [GtoPdb: 9]
Created with Highcharts 10.3.3ValuesChart context menu5-HT4 receptorpKd RatpKi RatpIC50 RatpEC50 RatpKd Guinea pigpKi Guinea pigpIC50 Guinea pigpEC50 Guinea pig024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT4 receptor in Rat [GtoPdb: 9] [UniProtKB: Q62758]
GtoPdb - - 9.3 pKd - - - Neuropharmacology (1997) 36: 671-9 [PMID:9225293]
5-HT4 receptor in Guinea pig [GtoPdb: 9]
GtoPdb - - 9.7 pKd 0.2 nM Kd Neuropharmacology (1997) 36: 671-9 [PMID:9225293]

ChEMBL data shown on this page come from version 34:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]