tamapin [Ligand Id: 2319] activity data from GtoPdb

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  • KCa2.1 in Human [GtoPdb: 381] [UniProtKB: Q92952]
Created with Highcharts 10.3.3ValuesChart context menuKCa2.1pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • KCa2.2 in Rat [GtoPdb: 382] [UniProtKB: P70604]
Created with Highcharts 10.3.3ValuesChart context menuKCa2.2pKd RatpKi RatpIC50 RatpEC50 Rat024681012Highcharts.com
  • KCa2.3 in Rat [GtoPdb: 383] [UniProtKB: P70605]
Created with Highcharts 10.3.3ValuesChart context menuKCa2.3pKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
KCa2.1 in Human [GtoPdb: 381] [UniProtKB: Q92952]
GtoPdb - - 7.4 pIC50 40 nM IC50 J Biol Chem (2002) 277: 46101-9 [PMID:12239213]
KCa2.2 in Rat [GtoPdb: 382] [UniProtKB: P70604]
GtoPdb - - 10.6 pIC50 - - - J Biol Chem (2002) 277: 46101-9 [PMID:12239213]
KCa2.3 in Rat [GtoPdb: 383] [UniProtKB: P70605]
GtoPdb - - 8.8 pIC50 - - - J Biol Chem (2002) 277: 46101-9 [PMID:12239213]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.