d[Cha4,Dab8]VP [Ligand Id: 2186] activity data from GtoPdb

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  • V1A receptor in Rat [GtoPdb: 366] [UniProtKB: P30560]
Created with Highcharts 10.3.3ValuesChart context menuV1A receptorpKd RatpKi RatpIC50 RatpEC50 Rat0123456Highcharts.com
  • V1B receptor in Rat [GtoPdb: 367] [UniProtKB: P48974]
Created with Highcharts 10.3.3ValuesChart context menuV1B receptorpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • V2 receptor in Rat [GtoPdb: 368] [UniProtKB: Q00788]
Created with Highcharts 10.3.3ValuesChart context menuV2 receptorpKd RatpKi RatpIC50 RatpEC50 Rat01234567Highcharts.com
  • OT receptor in Rat [GtoPdb: 369] [UniProtKB: P70536]
Created with Highcharts 10.3.3ValuesChart context menuOT receptorpKd RatpKi RatpIC50 RatpEC50 Rat02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
V1A receptor in Rat [GtoPdb: 366] [UniProtKB: P30560]
GtoPdb - - 5.4 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
V1B receptor in Rat [GtoPdb: 367] [UniProtKB: P48974]
GtoPdb - - 9.1 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
V2 receptor in Rat [GtoPdb: 368] [UniProtKB: Q00788]
GtoPdb - - 6.3 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
OT receptor in Rat [GtoPdb: 369] [UniProtKB: P70536]
GtoPdb - - 6.4 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.