spantide I [Ligand Id: 2096] activity data from GtoPdb

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  • NK1 receptor in Rabbit [GtoPdb: 360]
  • NK1 receptor in Rat [GtoPdb: 360] [UniProtKB: P14600]
  • NK1 receptor in Guinea pig [GtoPdb: 360]
Created with Highcharts 10.3.3ValuesChart context menuNK1 receptorpKd RabbitpKi RabbitpIC50 RabbitpEC50RabbitpA2 RabbitpKd RatpKi RatpIC50 RatpEC50 RatpA2 RatpKd GuineapigpKi GuineapigpIC50Guinea pigpEC50Guinea pigpA2 Guineapig0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
NK1 receptor in Rabbit [GtoPdb: 360]
GtoPdb - - 8.28 pIC50 5.2 nM IC50 Proc Natl Acad Sci USA (1990) 87: 4833-5 [PMID:1693780]
NK1 receptor in Rat [GtoPdb: 360] [UniProtKB: P14600]
GtoPdb - - 5.7 pIC50 2000 nM IC50 Life Sci (1984) 35: 1963-9 [PMID:6208451]
GtoPdb - - 5.6 pEC50 - - - Regul Pept (1990) 31: 75-82 [PMID:1702895]
NK1 receptor in Guinea pig [GtoPdb: 360]
GtoPdb - - 7.1 pA2 - - - Proc Natl Acad Sci USA (1990) 87: 4833-5 [PMID:1693780];
Regul Pept (1990) 31: 75-82 [PMID:1702895]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.