BIM 23068 [Ligand Id: 2040] activity data from GtoPdb

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  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
  • SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
Created with Highcharts 10.3.3ValuesChart context menuSST2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 Mouse024681012Highcharts.com
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
  • SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
  • SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
Created with Highcharts 10.3.3ValuesChart context menuSST3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 MousepKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
Created with Highcharts 10.3.3ValuesChart context menuSST4 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 8.8 pKi - - - Endocrinology (1994) 135: 2814-7 [PMID:7988476]
SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
GtoPdb - - 9.8 pIC50 - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 8.8 pKi - - - Endocrinology (1994) 135: 2814-7 [PMID:7988476]
SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
GtoPdb - - 9.1 pIC50 - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350]
SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
GtoPdb - - 8.4 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]
SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
GtoPdb - - 8 pKi - - - Endocrinology (1994) 135: 2814-7 [PMID:7988476]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.