[125I]LTT-SRIF-28 [Ligand Id: 2023] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
Created with Highcharts 10.3.3ValuesChart context menuSST1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
  • SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
Created with Highcharts 10.3.3ValuesChart context menuSST2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat024681012Highcharts.com
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
Created with Highcharts 10.3.3ValuesChart context menuSST3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
Created with Highcharts 10.3.3ValuesChart context menuSST4 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
  • SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
Created with Highcharts 10.3.3ValuesChart context menuSST5 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 Mouse024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
GtoPdb - - 8.8 pKd - - - Science (1998) 282: 737-40 [PMID:9784130]
GtoPdb - - 10 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 10 pKd - - - Science (1998) 282: 737-40 [PMID:9784130];
Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Eur J Pharmacol (1998) 348: 311-20 [PMID:9652348]
SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
GtoPdb - - 9.34 pKd 0.46 nM Kd Life Sci (1981) 28: 2191-8 [PMID:6114372];
Biochem Biophys Res Commun (1982) 105: 1538-45 [PMID:6125148]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 9.4 pKd - - - Science (1998) 282: 737-40 [PMID:9784130]
GtoPdb - - 10.3 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788];
FEBS Lett (1993) 321: 279-84 [PMID:8097479]
SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
GtoPdb - - 8.4 pKd - - - Science (1998) 282: 737-40 [PMID:9784130]
GtoPdb - - 9.6 pIC50 - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 9.2 pKd - - - Science (1998) 282: 737-40 [PMID:9784130]
GtoPdb - - 10.5 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
GtoPdb - - 11 pKd - - - Neuropharmacology (2000) 39: 1451-62 [PMID:10818261]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.