[125I]CGP 23996 [Ligand Id: 2022] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
There should be some charts here, you may need to enable JavaScript!
  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
There should be some charts here, you may need to enable JavaScript!
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
  • SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
There should be some charts here, you may need to enable JavaScript!
  • SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
There should be some charts here, you may need to enable JavaScript!
  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
  • SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
GtoPdb - - 9.6 pKd - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 9.8 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788];
Eur J Pharmacol (1998) 348: 311-20 [PMID:9652348]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 9.8 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
GtoPdb - - 9.4 pKd - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350]
SST4 receptor in Human [GtoPdb: 358] [UniProtKB: P31391]
GtoPdb - - 9.4 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 9.5 pKd - - - Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788];
Eur J Pharmacol (1998) 348: 311-20 [PMID:9652348]
SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
GtoPdb - - 9.8 pKd - - - Neuropharmacology (2000) 39: 1451-62 [PMID:10818261]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.