GPR61 inverse agonist 15 [Ligand Id: 14449] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GPR61 in Human [GtoPdb: 110] [UniProtKB: Q9BZJ8] | ||||||||
| GtoPdb | - | - | 9.68 | pKi | 0.21 | nM | Ki | J Med Chem (2026) 69: 7393-7404 [PMID:41834467] |
| GtoPdb | - | - | 8.21 | pIC50 | 6.2 | nM | IC50 | J Biol Chem (1998) 273: 15559-64 [PMID:9624146] |
| GPR61 in Mouse [GtoPdb: 110] [UniProtKB: Q8C010] | ||||||||
| GtoPdb | - | - | 9.14 | pKi | 0.72 | nM | Ki | J Med Chem (2026) 69: 7393-7404 [PMID:41834467] |
| GtoPdb | - | - | 7.7 | pIC50 | 20 | nM | IC50 | J Biol Chem (1998) 273: 15559-64 [PMID:9624146] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
