CHF6333 [Ligand Id: 14269] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • elastase, neutrophil expressed in Human [GtoPdb: 2358] [UniProtKB: P08246]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
elastase, neutrophil expressed in Human [GtoPdb: 2358] [UniProtKB: P08246]
GtoPdb Determined in a fluorescence hNE enzyme activity assay with peptide substrate MeOSuc-Ala-Ala-Pro-Val-AMC. - 7.7 pIC50 <20 nM IC50 US9828382B2. Pyrimidinone compounds as human neutrophil elastase inhibitors (2017)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.