MAP4 [Ligand Id: 1414] activity data from GtoPdb and ChEMBL
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
| ChEMBL ligand: CHEMBL1488784 |
|---|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mGlu4 receptor in Rat [GtoPdb: 292] [UniProtKB: P31423] | ||||||||
| GtoPdb | - | - | 4.6 | pKi | - | - | - | J Biol Chem (1999) 274: 10008-13 [PMID:10187777] |
| mGlu6 receptor in Rat [GtoPdb: 294] [UniProtKB: P35349] | ||||||||
| GtoPdb | - | - | 3.5 | pIC50 | - | - | - | Curr Drug Targets CNS Neurol Disord (2002) 1: 297-317 [PMID:12769621] |
| mGlu7 receptor in Human [GtoPdb: 295] [UniProtKB: Q14831] | ||||||||
| GtoPdb | - | - | 3.8 | pKi | - | - | - | Naunyn Schmiedebergs Arch Pharmacol (2000) 362: 546-54 [PMID:11138847] |
| mGlu8 receptor in Rat [GtoPdb: 296] [UniProtKB: P70579] | ||||||||
| GtoPdb | - | - | 7.6 | pIC50 | - | - | - |
Mol Pharmacol (1997) 51: 119-25 [PMID:9016353]; Brain Res Mol Brain Res (2000) 76: 180-90 [PMID:10719229] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
