casdatifan [Ligand Id: 13981] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| endothelial PAS domain protein 1 in Human [GtoPdb: 3148] [UniProtKB: Q99814] | ||||||||
| GtoPdb | Measuring inhibition of HIF-2α-mediated VEGF secretion by 786-O cell (as a proxy for HIF-2α-mediated gene transcription) | - | 7.54 | pIC50 | 28.9 | nM | IC50 | Br J Pharmacol (2025) 182: 4147-4167 [PMID:40400177] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
