PARP1 inhibitor (S)-G9 [Ligand Id: 13961] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • poly(ADP-ribose) polymerase 1 in Human [GtoPdb: 2771] [UniProtKB: P09874]
There should be some charts here, you may need to enable JavaScript!
  • poly(ADP-ribose) polymerase 2 in Human [GtoPdb: 2772] [UniProtKB: Q9UGN5]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
poly(ADP-ribose) polymerase 1 in Human [GtoPdb: 2771] [UniProtKB: P09874]
GtoPdb - - 9.72 pIC50 0.19 nM IC50 J Med Chem (2025) :
poly(ADP-ribose) polymerase 2 in Human [GtoPdb: 2772] [UniProtKB: Q9UGN5]
GtoPdb - - 7.59 pIC50 26 nM IC50 J Med Chem (2025) :

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.