EOS-984 [Ligand Id: 13932] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Equilibrative nucleoside transporter 1 in Human [GtoPdb: 1117] [UniProtKB: Q99808] | ||||||||
| GtoPdb | Binned IC50 value, determined in a fluorescent competition binding assay using JAR cells expressing ENT1 | - | 9 | pIC50 | 1 | nM | IC50 | US20230203058A1. Macrocyclic diamine derivatives as ent inhibitors for the treatment of cancers, and combination thereof with adenosine receptor antagonists (2023) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
