EB-42168 [Ligand Id: 13903] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| leucine rich repeat kinase 2 in Human [GtoPdb: 2059] [UniProtKB: Q5S007] | ||||||||
| GtoPdb | Measuring inhibition of pS935-LRRK2 (WT) in a FRET assay | - | 6.84 | pIC50 | 145 | nM | IC50 | J Med Chem (2020) 63: 14821-14839 [PMID:33197196] |
| GtoPdb | Measuring inhibition of pS935-LRRK2 (G2019S) in a FRET assay | - | 8.96 | pIC50 | 1.1 | nM | IC50 | J Med Chem (2020) 63: 14821-14839 [PMID:33197196] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
