claturafenib [Ligand Id: 13808] activity data from GtoPdb

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  • B-Raf proto-oncogene, serine/threonine kinase in Human [GtoPdb: 1943] [UniProtKB: P15056]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
B-Raf proto-oncogene, serine/threonine kinase in Human [GtoPdb: 1943] [UniProtKB: P15056]
GtoPdb Dimer stability determined in an isothermal stability shift assay using lysate from cells expressing BRAFV600E. - 7.46 pEC50 34.4 nM EC50 Cancer Discov (2024) 14: 1599-1611 [PMID:38691346]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.