retatrutide [Ligand Id: 13769] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| GIP receptor in Human [GtoPdb: 248] [UniProtKB: P48546] | ||||||||
| GtoPdb | - | - | 10.24 | pKi | 0.06 | nM | Ki | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
| GtoPdb | Determined in a cAMP assay | - | 10.19 | pEC50 | 0.06 | nM | EC50 | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
| GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220] | ||||||||
| GtoPdb | - | - | 8.14 | pKi | 7.2 | nM | Ki | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
| GtoPdb | Determined in a cAMP assay | - | 9.11 | pEC50 | 0.78 | nM | EC50 | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
| glucagon receptor in Human [GtoPdb: 251] [UniProtKB: P47871] | ||||||||
| GtoPdb | - | - | 8.25 | pKi | 5.6 | nM | Ki | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
| GtoPdb | Determined in a cAMP assay | - | 8.24 | pEC50 | 5.79 | nM | EC50 | Cell Metab (2022) 34: 1234-1247.e9 [PMID:35985340] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
