SH-1028 [Ligand Id: 13760] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of wild type EGFR | - | 7.74 | pIC50 | 18 | nM | IC50 | Front Pharmacol (2021) 12: 665253 [PMID:33986687] |
| GtoPdb | Inhibition of EGFRL858R | - | 9.15 | pIC50 | 0.7 | nM | IC50 | Front Pharmacol (2021) 12: 665253 [PMID:33986687] |
| GtoPdb | Inhibition of EGFRL858R/T790M | - | 10 | pIC50 | 0.1 | nM | IC50 | Front Pharmacol (2021) 12: 665253 [PMID:33986687] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
