Lu AF64196 [Ligand Id: 13576] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • phosphodiesterase 1A in Human [GtoPdb: 1294] [UniProtKB: P54750]
There should be some charts here, you may need to enable JavaScript!
  • phosphodiesterase 1B in Human [GtoPdb: 1295] [UniProtKB: Q01064]
There should be some charts here, you may need to enable JavaScript!
  • phosphodiesterase 1C in Human [GtoPdb: 1296] [UniProtKB: Q14123]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
phosphodiesterase 1A in Human [GtoPdb: 1294] [UniProtKB: P54750]
GtoPdb - - 7.24 pKi 57.5 nM Ki Br J Pharmacol (2017) 174: 4186-4198 [PMID:28910498]
phosphodiesterase 1B in Human [GtoPdb: 1295] [UniProtKB: Q01064]
GtoPdb - - 7.86 pKi 13.8 nM Ki Br J Pharmacol (2017) 174: 4186-4198 [PMID:28910498]
phosphodiesterase 1C in Human [GtoPdb: 1296] [UniProtKB: Q14123]
GtoPdb - - 7.33 pKi 46.8 nM Ki Br J Pharmacol (2017) 174: 4186-4198 [PMID:28910498]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.