compound 43 [PMID: 34781683] [Ligand Id: 13359] activity data from GtoPdb

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  • HCA2 receptor in Human [GtoPdb: 312] [UniProtKB: Q8TDS4]
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  • coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
HCA2 receptor in Human [GtoPdb: 312] [UniProtKB: Q8TDS4]
GtoPdb - - 7.4 pEC50 39.8 nM EC50 Pharmacology Research & Perspectives (2024) :
coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55]
GtoPdb Inhibitor potency vs. enzyme activity. - 5.43 pIC50 3700 nM IC50 J Med Chem (2021) 64: 16650-16674 [PMID:34781683]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.